Recently, we reported that the TM2 peptide analogue shows the pharmacological behaviour of a competitive antagonist for β-arrestin 2 recruitment to ACKR3-Tango upon agonist stimulation, whereas the TM7 peptide analogue was inactive; the TM4 peptide exhibited a behaviour similar to the TM2 peptide, but this effect did not reach statistical significance [ 21 ].
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Identification and functional characterization of arginine vasopressin receptor 1A : atypical chemokine receptor 3 heteromers in vascular smooth muscle.
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